Design, synthesis and molecular docking of novel diarylcyclohexenone and diarylindazole derivatives as tubulin polymerization inhibitors
Author:
Affiliation:
1. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Nahda University in Beni Suef, Kornish Al Nile, Beni Suef, Egypt;
2. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo, Egypt
Publisher
Informa UK Limited
Subject
Drug Discovery,Pharmacology,General Medicine
Link
https://www.tandfonline.com/doi/pdf/10.1080/14756366.2016.1244532
Reference21 articles.
1. Pharmacophore Modeling, Atom based 3D-QSAR and Docking Studies of Chalcone derivatives as Tubulin inhibitors
2. An Overview of Tubulin Inhibitors That Interact with the Colchicine Binding Site
3. Combined Molecular Docking, 3D-QSAR, and Pharmacophore Model: Design of Novel Tubulin Polymerization Inhibitors by Binding to Colchicine-binding Site
4. Interaction of colchicine analogues with purified tubulin
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