Efficient One-Pot Synthesis of the GABAB Positive Allosteric Modulator (R,S)-5,7-Di-tert-butyl-3-hydroxy-3-trifluoromethyl-3H-benzofuran-2-one-Reference-Cited by-同舟云学术

Efficient One-Pot Synthesis of the GABAB Positive Allosteric Modulator (R,S)-5,7-Di-tert-butyl-3-hydroxy-3-trifluoromethyl-3H-benzofuran-2-one

Published:2008-09-29 Issue:20 Volume:38 Page:3398-3405
ISSN:0039-7911
Container-title:Synthetic Communications
language:en
Short-container-title:Synthetic Communications

Author:

Alker Andre M.¹,Grillet François¹,Malherbe Pari¹,Norcross Roger D.¹,Thomas Andrew W.¹,Masciadri Raffaello¹

Affiliation:

1. a Hoffmann-La Roche AG , Basel, Switzerland

Publisher

Informa UK Limited

Subject

Organic Chemistry

Link

https://www.tandfonline.com/doi/pdf/10.1080/00397910801979403

Reference13 articles.

1. Dyachenko , V. I. Galakhov , M. V. Kolomiets , A. F. Fokin , A. V. Steric effects of ortho substituents in reactions of phenols and phenolates with polyfluoro ketones . Izvestiya Akademii Nauk SSSR, Ser. Khim . 1989 , 923 – 928 .

2. Unusual Friedel–Crafts reactions. Part 7. Synthesis of α-(2-hydroxyphenyl)ethyl lactates and their reductive cyclization to 3-methyl-2,3-dihydrobenzofuran-2-ols

3. A Facile and Efficient Synthesis of (o-Hydroxyaryl)-glycolic Acid Derivatives

4. Catalytic, Highly Enantioselective Friedel−Crafts Reactions of Aromatic and Heteroaromatic Compounds to Trifluoropyruvate. A Simple Approach for the Formation of Optically Active Aromatic and Heteroaromatic Hydroxy Trifluoromethyl Esters

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