The Allosteric Modulation of the GABAB Receptor: A Medicinal Chemistry Perspective
Author:
Publisher
Springer International Publishing
Link
http://link.springer.com/content/pdf/10.1007/978-3-319-46044-4_3
Reference71 articles.
1. Abraham, N., & Goldman, H. B. (2015). An update on the pharmacology for the lower urinary tract dysfunction. Expert Opinion on Pharmacotherapy, 16, 79–93.
2. Adams, C. L., & Lawrence, A. J. (2007). CGP7930: a positive allosteric modulator of the GABAB receptor. CNS Drug Reviews, 13, 308–316.
3. Agabio, R., & Colombo, G. (2014). GABAB receptor ligands for the treatment of alcohol use disorder: Preclinical and clinical evidence. Frontiers in Neuroscience, 8, 140.
4. Alker, A. M., Grillet, F., Malherbe, P., Norcross, R. D., Thomas, A. W., & Masciadri, R. (2008). Efficient one-pot synthesis of the GABAB positive allosteric modulator (R, S)-5,7-di-tert-butyl-3-hydroxy-3-trifluoromethyl-3H-benzofuran-2-one. Synthetic Communications, 38, 3398–3405.
5. Balerio, G. N., & Rubio, M. C. (2002). Baclofen analgesia: Involvement of the GABAergic system. Pharmacological Research, 46, 281–286.
Cited by 12 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Synthesis of R–GABA Derivatives via Pd(II) Catalyzed Enantioselective C(sp3)−H Arylation and Virtual Validation with GABAB1 Receptor for Potential leads;Chemistry – An Asian Journal;2024-05-06
2. Positive allosteric modulators of the GABAB receptor: a new class of ligands with therapeutic potential for alcohol use disorder;Alcohol and Alcoholism;2024-03-16
3. The Novel Positive Allosteric Modulator of the GABAB Receptor, KK-92A, Suppresses Alcohol Self-Administration and Cue-Induced Reinstatement of Alcohol Seeking in Rats;Frontiers in Cell and Developmental Biology;2021-10-28
4. COR758, a negative allosteric modulator of GABAB receptors;Neuropharmacology;2021-05
5. The GABAB receptor positive allosteric modulator COR659: In vitro metabolism, in vivo pharmacokinetics in rats, synthesis and pharmacological characterization of metabolically protected derivatives;European Journal of Pharmaceutical Sciences;2020-12
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3