Three-step synthetic procedure to prepare dolutegravir, cabotegravir, and bictegravir
Author:
Affiliation:
1. Department of Medicinal Chemistry, Zunyi Medical University, Zunyi, People’s Republic of China
2. Department of Pharmaceutical Analysis, Zunyi Medical University, Zunyi, People’s Republic of China
Funder
Key Project of Guizhou Provincial Administration of Traditional Chinese Medicine
Joint Funds of Zunyi City
Guizhou Provincial Administration of Traditional Chinese Medicine
Science and Technology Foundation of Guizhou Province
Publisher
Informa UK Limited
Subject
Environmental Chemistry,General Chemistry
Link
https://www.tandfonline.com/doi/pdf/10.1080/17518253.2022.2057200
Reference17 articles.
1. The inhibition process of HIV-1 integrase by diketoacids molecules: Understanding the factors governing the better efficiency of dolutegravir
2. Pharmacokinetics of Dolutegravir in a Premature Neonate after HIV Treatment Intensification during Pregnancy
3. Successful prevention of HIV mother-to-child transmission with dolutegravir-based combination antiretroviral therapy in a vertically infected pregnant woman with multiclass highly drug-resistant HIV-1
4. Structure-Guided Optimization of HIV Integrase Strand Transfer Inhibitors
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