Synthetic Approaches to a Key Pyridone-carboxylic Acid Precursor Common to the HIV-1 Integrase Strand Transfer Inhibitors Dolutegravir, Bictegravir, and Cabotegravir-Reference-Cited by-同舟云学术

Synthetic Approaches to a Key Pyridone-carboxylic Acid Precursor Common to the HIV-1 Integrase Strand Transfer Inhibitors Dolutegravir, Bictegravir, and Cabotegravir

Published:2023-04-20 Issue:5 Volume:27 Page:847-853
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Mahajan Pankaj S.¹,Burke Terrence R.¹

Affiliation:

1. Chemical Biology Laboratory, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Frederick, Maryland 21702, United States

Funder

National Cancer Institute

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.3c00063

Reference28 articles.

1. HIV Fact Sheet. World Health Organization, November 9, 2022. https://www.who.int/news-room/fact-sheets/detail/hiv-aids (accessed 2023-02-14).

2. Human Immunodeficiency Virus/AIDS in the Era of Coronavirus Disease 2019: A Juxtaposition of 2 Pandemics

3. Update and latest advances in antiretroviral therapy

4. New designs for HIV-1 integrase inhibitors: a patent review (2018-present)

5. Retroviral DNA Integration

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