Structure-Guided Optimization of HIV Integrase Strand Transfer Inhibitors-Reference-Cited by-同舟云学术

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Structure-Guided Optimization of HIV Integrase Strand Transfer Inhibitors

Published:2017-08-10 Issue:17 Volume:60 Page:7315-7332
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Zhao Xue Zhi,Smith Steven J.,Maskell Daniel P.¹,Métifiot Mathieu²,Pye Valerie E.¹,Fesen Katherine²,Marchand Christophe²,Pommier Yves²,Cherepanov Peter¹³,Hughes Stephen H.²,Burke Terrence R.^ORCID

Affiliation:

1. Chromatin Structure and Mobile DNA, The Francis Crick Institute, London NW1 1AT, United Kingdom

2. Developmental Therapeutics Branch and Laboratory of Molecular Pharmacology, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland 20892, United States

3. Imperial College London, St-Mary’s Campus, Norfolk Place, London W2 1PG, United Kingdom

Funder

National Cancer Institute

NIH Office of the Director

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

http://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b00596

Reference51 articles.

1. Retroviral DNA Integration

2. Discovery of Raltegravir, a Potent, Selective Orally Bioavailable HIV-Integrase Inhibitor for the Treatment of HIV-AIDS Infection

3. Novel HIV-1 Integrase Inhibitors Derived from Quinolone Antibiotics

4. Carbamoyl Pyridone HIV-1 Integrase Inhibitors 3. A Diastereomeric Approach to Chiral Nonracemic Tricyclic Ring Systems and the Discovery of Dolutegravir (S/GSK1349572) and (S/GSK1265744)

5. Inhibitors of Strand Transfer That Prevent Integration and Inhibit HIV-1 Replication in Cells

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5. N-Substituted Bicyclic Carbamoyl Pyridones: Integrase Strand Transfer Inhibitors that Potently Inhibit Drug-Resistant HIV-1 Integrase Mutants;ACS Infectious Diseases;2024-02-12

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