Predictive QSAR workflow for the in silico identification and screening of novel HDAC inhibitors-Reference-Cited by-同舟云学术

Predictive QSAR workflow for the in silico identification and screening of novel HDAC inhibitors

Published:2009-02-10 Issue:3 Volume:13 Page:301-311
ISSN:1381-1991
Container-title:Molecular Diversity
language:en
Short-container-title:Mol Divers

Author:

Melagraki Georgia,Afantitis Antreas,Sarimveis Haralambos,Koutentis Panayiotis A.,Kollias George,Igglessi-Markopoulou Olga

Publisher

Springer Science and Business Media LLC

Subject

Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Drug Discovery,Molecular Biology,General Medicine,Information Systems,Catalysis

Link

http://link.springer.com/content/pdf/10.1007/s11030-009-9115-2.pdf

Reference58 articles.

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2. Elaut G, Rogiers V, Vanhaecke T (2007) The pharmaceutical potential of histone deacetylase inhibitors. Curr Pharm Des 13: 2584–2620. doi: 10.2174/138161207781663064

3. An W (2007) Histone acetylation and methylation: combinatorial players for transcriptional regulation. Subcell Biochem 41: 351–369

4. de Ruijter AJM, van Gennip AH, Caron HN, Kemp S, van Kuilenburg ABP (2003) Histone deacetylases (HDACs): characterization of the classical HDAC family. Biochem J 370: 737–749. doi: 10.1042/BJ20021321

5. Rasheed WK, Johnstone RW, Prince HM (2007) Histone deacetylase inhibitors in cancer therapy. Expert Opin Investig Drugs 16: 659–678. doi: 10.1517/13543784.16.5.659

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