Covalent Kinase Inhibitors: An Overview
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Publisher
Springer International Publishing
Link
http://link.springer.com/content/pdf/10.1007/7355_2020_103
Reference142 articles.
1. Singh J, Petter RC, Baillie TA, Whitty A (2011) The resurgence of covalent drugs. Nat Rev Drug Discov 10:307–317. https://doi.org/10.1038/nrd3410
2. Bauer RA (2015) Covalent inhibitors in drug discovery: from accidental discoveries to avoided liabilities and designed therapies. Drug Discov Today 20:1061–1073. https://doi.org/10.1016/j.drudis.2015.05.005
3. Baillie TA (2016) Targeted covalent inhibitors for drug design. Angew Chem Int Ed 55:13408–13421. https://doi.org/10.1002/anie.201601091
4. Singh J, Petter RC, Kluge AF (2010) Targeted covalent drugs of the kinase family. Curr Opin Chem Biol 14:475–480. https://doi.org/10.1016/j.cbpa.2010.06.168
5. Barf T, Kaptein A (2012) Irreversible protein kinase inhibitors: balancing the benefits and risks. J Med Chem 55:6243–6262. https://doi.org/10.1021/jm3003203
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