Small Quaternary Inhibitors K298 and K524: Cholinesterases Inhibition, Absorption, Brain Distribution, and Toxicity-Reference-Cited by-同舟云学术

Small Quaternary Inhibitors K298 and K524: Cholinesterases Inhibition, Absorption, Brain Distribution, and Toxicity

Published:2015-12-08 Issue:2 Volume:29 Page:267-274
ISSN:1029-8428
Container-title:Neurotoxicity Research
language:en
Short-container-title:Neurotox Res

Author:

Karasova Jana Zdarova,Hroch Milos,Musilek Kamil,Kuca Kamil

Funder

Ministry of Defense (CZ)

University Hospital in Hradec Kralove (CZ)

University of Hradec Kralove (CZ)

Publisher

Springer Science and Business Media LLC

Subject

Toxicology,General Neuroscience

Link

http://link.springer.com/content/pdf/10.1007/s12640-015-9582-4.pdf

Reference27 articles.

1. Amourette C, Lamproglou I, Barbier L, Fauquette W, Zoppe A, Viret R et al (2009) Gulf war illness: effects of repeated stress and pyridostigmine treatment on blood-brain barrier permeability and cholinesterase activity in rat brain. Behav Brain Res 203(2):207–214

2. Arning J, Stolte S, Boschen A, Stock F, Pitner WR, Welz-Biermann U et al (2008) Qualitative and quantitative structure activity relationships for the inhibitory effects of cationic head groups, functionalised side chains and anions of ionic liquids on acetylcholinesterase. Green Chem 10(1):47–58

3. Chernikova EY, Fedorov YV, Fedorova OA (2012) Cucurbituril as a new “host” of organic molecules in inclusion complexes. Russ Chem B 61(7):1363–1390

4. Conejo-Garcia A, Pisani L, Nunez MDC, Catto M, Nicolotti O, Leonetti F et al (2011) Homodimeric bis-quaternary heterocyclic ammonium salts as potent acetyl- and butyrylcholinesterase inhibitors: a systematic investigation of the influence of linker and cationic heads over affinity and selectivity. J Med Chem 54(8):2627–2645

5. Foy DS, Trepanier LA, Shelton GD (2011) Cholinergic crisis after neostigmine administration in a dog with acquired focal myasthenia gravis. J Vet Emerg Crit Car 21(5):547–551

Cited by 10 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Determination of K869, a Novel Oxime Reactivator of Acetylcholinesterase, in Rat Body Fluids and Tissues by Liquid-Chromatography Methods: Pharmacokinetic Study;Journal of Pharmaceutical Sciences;2021-04

2. Indol-2-Carboxylic Acid Esters Containing N-Phenylpiperazine Moiety - Preparation and Cholinesterase-inhibiting Activity;Current Organic Synthesis;2020-10-28

3. Donepezil and Rivastigmine: Pharmacokinetic Profile and Brain-targeting After Intramuscular Administration in Rats;IRAN J PHARM RES;2020

4. UHPLC-HRMS study of anti-Alzheimer’s drug candidates: metabolism of 7-MEOTA-tryptophan hybrids hampers their passage into brain;Journal of Pharmaceutical and Biomedical Analysis;2019-09

5. 1-Benzyl-4-methylpiperidinyl moiety in donepezil: The priority ticket across the blood-brain-barrier in rats;Journal of Chromatography B;2018-08