[18F]BTK-1: A Novel Positron Emission Tomography Tracer for Imaging Bruton’s Tyrosine Kinase-Reference-Cited by-同舟云学术

[18F]BTK-1: A Novel Positron Emission Tomography Tracer for Imaging Bruton’s Tyrosine Kinase

Published:2022-04-28 Issue:5 Volume:24 Page:830-841
ISSN:1536-1632
Container-title:Molecular Imaging and Biology
language:en
Short-container-title:Mol Imaging Biol

Author:

Skaddan Marc B.,Wooten Dustin W.,Wilcox Kyle C.,Voorbach Martin J.,Reuter David R.,Jia Zhaozhong J.,Foster-Duke Kelly D.,Hickson Jonathan A.,Vaidyanathan Srirajan,Reed Aimee D.,Tovcimak Ann E.,Guo Qi,Comley Robert A.,Lee Lance,Finnema Sjoerd J.,Mudd Sarah R.^ORCID

Publisher

Springer Science and Business Media LLC

Subject

Cancer Research,Radiology, Nuclear Medicine and imaging,Oncology

Link

https://link.springer.com/content/pdf/10.1007/s11307-022-01733-1.pdf

Reference22 articles.

1. Burger JA, Wiestner A (2018) Targeting B cell receptor signalling in cancer: preclinical and clinical advances. Nat Rev Cancer 18:148–167

2. Pal Singh S, Dammeijer F, Hendriks RW (2018) Role of Bruton’s tyrosine kinase in B cells and malignancies. Mol Cancer 17:57

3. Lucas F, Woyach JA (2019) Inhibiting Bruton’s Tyrosine Kinase in CLL and Other B-Cell Malignancies. Target Oncol 14:125–138

4. Jacobs L, Habringer S, Slawska J et al (2017) Functional imaging in combination with mutation status aids prediction of response to inhibiting B-cell receptor signaling in lymphoma. Oncotarget 8:78917–78929

5. Dahl K, Turner T, Vasdev N (2020) Radiosynthesis of a Bruton’s tyrosine kinase inhibitor, [(11) C]Tolebrutinib, via palladium-NiXantphos-mediated carbonylation. J Label Compd Radiopharm 63:482–487

Cited by 4 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Labeling of Bruton’s Tyrosine Kinase (BTK) Inhibitor [11C]BIO-2008846 in Three Different Positions and Measurement in NHP Using PET;International Journal of Molecular Sciences;2024-07-18

2. Preliminary PET imaging of [¹¹C]evobrutinib in mouse models of colorectal cancer, SARS‐CoV‐2, and lung damage: Radiosynthesis via base‐aided palladium‐NiXantphos‐mediated¹¹C‐carbonylation;Journal of Labelled Compounds and Radiopharmaceuticals;2023-09-10

3. Synthesis and Preclinical Evaluation of a Novel Fluorine-18-Labeled Tracer for Positron Emission Tomography Imaging of Bruton’s Tyrosine Kinase;ACS Pharmacology & Translational Science;2023-02-10

4. Pipeline Impact of Radiolabeled Compounds in Drug Discovery and Development;ACS Medicinal Chemistry Letters;2022-09-16