Mechanistic and Structural Features of PROTAC Ternary Complexes
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Publisher
Springer US
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https://link.springer.com/content/pdf/10.1007/978-1-0716-1665-9_5
Reference85 articles.
1. Hill AV (1910) The possible effects of the aggregation of the molecules of haemoglobin on its dissociation curves. J Physiol Lond 40:4–7
2. Labrijn AF, Janmaat ML, Reichert JM, Parren P (2019) Bispecific antibodies: a mechanistic review of the pipeline. Nat Rev Drug Discov 18(8):585–608. https://doi.org/10.1038/s41573-019-0028-1
3. Profit AA, Lee TR, Lawrence DS (1999) Bivalent inhibitors of protein tyrosine kinases. J Am Chem Soc 121(2):280–283. https://doi.org/10.1021/ja983515n
4. Tanaka M, Roberts JM, Seo HS, Souza A, Paulk J, Scott TG, DeAngelo SL, Dhe-Paganon S, Bradner JE (2016) Design and characterization of bivalent BET inhibitors. Nat Chem Biol 12(12):1089–1096. https://doi.org/10.1038/Nchembio.2209
5. Waring MJ, Chen HW, Rabow AA, Walker G, Bobby R, Boiko S, Bradbury RH, Callis R, Clark E, Dale I, Daniels DL, Dulak A, Flavell L, Holdgate G, Jowitt TA, Kikhney A, McAlister M, Mendez J, Ogg D, Patel J, Petteruti P, Robb GR, Robers MB, Saif S, Stratton N, Svergun DI, Wang WX, Whittaker D, Wilson DM, Yao Y (2016) Potent and selective bivalent inhibitors of BET bromodomains. Nat Chem Biol 12(12):1097–1104. https://doi.org/10.1038/Nchembio.2210
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