Mechanistic and Structural Features of PROTAC Ternary Complexes
Author:
Publisher
Springer US
Link
https://link.springer.com/content/pdf/10.1007/978-1-0716-1665-9_5
Reference85 articles.
1. Hill AV (1910) The possible effects of the aggregation of the molecules of haemoglobin on its dissociation curves. J Physiol Lond 40:4–7
2. Labrijn AF, Janmaat ML, Reichert JM, Parren P (2019) Bispecific antibodies: a mechanistic review of the pipeline. Nat Rev Drug Discov 18(8):585–608. https://doi.org/10.1038/s41573-019-0028-1
3. Profit AA, Lee TR, Lawrence DS (1999) Bivalent inhibitors of protein tyrosine kinases. J Am Chem Soc 121(2):280–283. https://doi.org/10.1021/ja983515n
4. Tanaka M, Roberts JM, Seo HS, Souza A, Paulk J, Scott TG, DeAngelo SL, Dhe-Paganon S, Bradner JE (2016) Design and characterization of bivalent BET inhibitors. Nat Chem Biol 12(12):1089–1096. https://doi.org/10.1038/Nchembio.2209
5. Waring MJ, Chen HW, Rabow AA, Walker G, Bobby R, Boiko S, Bradbury RH, Callis R, Clark E, Dale I, Daniels DL, Dulak A, Flavell L, Holdgate G, Jowitt TA, Kikhney A, McAlister M, Mendez J, Ogg D, Patel J, Petteruti P, Robb GR, Robers MB, Saif S, Stratton N, Svergun DI, Wang WX, Whittaker D, Wilson DM, Yao Y (2016) Potent and selective bivalent inhibitors of BET bromodomains. Nat Chem Biol 12(12):1097–1104. https://doi.org/10.1038/Nchembio.2210
Cited by 41 articles. 订阅此论文施引文献 订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献
1. Mechanistic insights into a heterobifunctional degrader-induced PTPN2/N1 complex;Communications Chemistry;2024-08-16
2. BCR::ABL1 Proteolysis-targeting chimeras (PROTACs): The new frontier in the treatment of Ph+ leukemias?;Leukemia;2024-08-04
3. Targeted Protein Degradation: Current and Emerging Approaches for E3 Ligase Deconvolution;Journal of Medicinal Chemistry;2024-07-09
4. A CRISPR activation screen identifies FBXO22 supporting targeted protein degradation;Nature Chemical Biology;2024-07-04
5. Ultrasound-Activated PROTAC Prodrugs Overcome Immunosuppression to Actuate Efficient Deep-Tissue Sono-Immunotherapy in Orthotopic Pancreatic Tumor Mouse Models;Nano Letters;2024-07-02
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3