Unravelling the Mechanistic Role of Quinazolinone Pharmacophore in the Inhibitory Activity of Bis-quinazolinone Derivative on Tankyrase-1 in the Treatment of Colorectal Cancer (CRC) and Non-small Cell Lung Cancer (NSCLC): A Computational Approach-Reference-Cited by-同舟云学术

Unravelling the Mechanistic Role of Quinazolinone Pharmacophore in the Inhibitory Activity of Bis-quinazolinone Derivative on Tankyrase-1 in the Treatment of Colorectal Cancer (CRC) and Non-small Cell Lung Cancer (NSCLC): A Computational Approach

Published:2021-08-28 Issue: Volume: Page:
ISSN:1085-9195
Container-title:Cell Biochemistry and Biophysics
language:en
Short-container-title:Cell Biochem Biophys

Author:

Okunlola Felix O.,Akawa Oluwole B.,Subair Temitayo I.,Omolabi Kehinde F.,Soliman Mahmoud E. S.^ORCID

Publisher

Springer Science and Business Media LLC

Subject

Cell Biology,Biochemistry,General Medicine,Biophysics

Link

https://link.springer.com/content/pdf/10.1007/s12013-021-01027-3.pdf

Reference69 articles.

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2. Tomassi, S., et al. (2020). From PARP1 to TNKS2 inhibition: a structure-based approach. ACS Medicinal Chemistry Letters, 11(5), 862–868. https://doi.org/10.1021/acsmedchemlett.9b00654.

3. Hottiger, M. O., Hassa, P. O., Lüscher, B., Schüler, H., & Koch-Nolte, F. (2010). Toward a unified nomenclature for mammalian ADP-ribosyltransferases. Trends in Biochemical Sciences, 35(4), 208–219. https://doi.org/10.1016/j.tibs.2009.12.003.

4. Langelier, M. F., Eisemann, T., Riccio, A. A., & Pascal, J. M. (2018). PARP family enzymes: regulation and catalysis of the poly(ADP-ribose) posttranslational modification. Current Opinion in Structural Biology, 53, 187–198. https://doi.org/10.1016/j.sbi.2018.11.002.

5. Palazzo, L., Mikoc, A., & Ahel, I. (2018). ADP-RIBOSYLATION: new facets of an ancient modification. The FEBS Journal, 284(18), 2932–2946. https://doi.org/10.1111/ijlh.12426.

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