Development of Novel Dual Binders as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors-Reference-Cited by-同舟云学术

Development of Novel Dual Binders as Potent, Selective, and Orally Bioavailable Tankyrase Inhibitors

Published:2013-12-11 Issue:24 Volume:56 Page:10003-10015
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hua Zihao¹,Bregman Howard¹,Buchanan John L.¹,Chakka Nagasree¹,Guzman-Perez Angel¹,Gunaydin Hakan¹,Huang Xin¹,Gu Yan¹,Berry Virginia¹,Liu Jingzhou¹,Teffera Yohannes¹,Huang Liyue¹,Egge Bryan¹,Emkey Renee¹,Mullady Erin L.¹,Schneider Steve¹,Andrews Paul S.¹,Acquaviva Lisa¹,Dovey Jennifer¹,Mishra Ankita¹,Newcomb John¹,Saffran Douglas¹,Serafino Randy¹,Strathdee Craig A.¹,Turci Susan M.¹,Stanton Mary¹,Wilson Cindy¹,DiMauro Erin F.¹

Affiliation:

1. Department of Chemistry Research and Discovery, ‡Department of Pharmacokinetics and Drug Metabolism, §Oncology Research, ∥Department of Molecular Structure, ⊥Bioassay and Profiling, and #Pharmaceutics, Amgen Inc., 360 Binney Street, Cambridge, Massachusetts 02142, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm401317z

Reference31 articles.

1. Wnt/β-Catenin Signaling in Development and Disease

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