Enzymatic Synthesis of 2′-O-acyl Prodrugs of 1-(β-D-arabinofuranosyl)-5(E)-(2-bromovinyl)uracil and of 2′-O-acyl-araU, -araC and -araA
Author:
Affiliation:
1. Dipartimento di Scienze Farmaceutiche, Università di Ferrara, Via Fossato, di Mortara 17-19, 1-44100 Ferrara, Italy
2. R&D Division, Yamasa Corporation, 10–1, Araoicho 2 Chome, Choshi, Chiba-ken 288, Japan
Abstract
Publisher
SAGE Publications
Link
http://journals.sagepub.com/doi/pdf/10.1177/095632029800900103
Reference21 articles.
1. New Antiherpesvirus Agents
2. Prodrugs of 9-(.beta.-D-arabinofuranosyl)adenine. 2. Synthesis and evaluation of a number of 2',3'- and 3',5'-di-O-acyl derivatives
3. Facile access to 2′-O-acyl prodrugs of 1- (β-d-arabinofuranosyl)-5(E)-(2-bromovinyl)uracil (BVAraU) via regioselective esterase-catalyzed hydrolysis of 2′ 3′, 5′-triesters1
4. Selective O-acylation. Preparation of 1-(2,3,5-tri-O-acetyl-β-D-arabino-pentofuranosyl)cytosine hydrochloride
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1. Enzymatic regioselective and complete deacetylation of two arabinonucleosides;Journal of Molecular Catalysis B: Enzymatic;2010-03
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