Non-regioselective functionalization: an underestimate chemical diversity generator in medicinal chemistry
Author:
Affiliation:
1. Chemistry Research & Drug Design, Chiesi Farmaceutici S.p.A, Centro Ricerche, Largo Belloli 11/a, Parma 43122, Italy
Publisher
Future Science Ltd
Subject
Drug Discovery,Pharmacology,Molecular Medicine
Link
https://www.future-science.com/doi/pdf/10.4155/fmc-2021-0011
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1. Estimation of clinical trial success rates and related parameters
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4. Diversity-oriented synthesis; a challenge for synthetic chemistsElectronic supplementary information (ESI) available: Excel file of all the FDA new molecular entities between the years 1998 and July 2003, and new drug approvals between the years 1990 and 2002. See http://www.rsc.org/suppdata/ob/b3/b310752n/
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