Conference Report: G-protein coupled receptor and kinase targets: advances in drug discovery from molecular to clinical-Reference-Cited by-同舟云学术

Conference Report: G-protein coupled receptor and kinase targets: advances in drug discovery from molecular to clinical

Published:2011-07 Issue:9 Volume:3 Page:1097-1100
ISSN:1756-8919
Container-title:Future Medicinal Chemistry
language:en
Short-container-title:Future Medicinal Chemistry

Author:

Spencer John¹

Affiliation:

1. School of Science, University of Greenwich at Medway, Chatham, Kent, ME4 4TB, UK.

Abstract

The conference was organized by Visiongain and focused on a number of industrially relevant advances in G-protein coupled receptor and kinase research. Commercial stands were provided by Genscript (Bioassays), Merck Millipore (profiling services), Schrödinger (modeling) and Corning (assay development). The overall attendance was approximately 40 delegates taking part in four sessions over the two days.

Publisher

Future Science Ltd

Subject

Drug Discovery,Pharmacology,Molecular Medicine

Link

http://www.future-science.com/doi/pdf/10.4155/fmc.11.78

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2. Drug Design for G-Protein-Coupled Receptors by a Ligand-Based NMR Method

3. Selective inhibition of BET bromodomains

4. β‐Galactosidase enzyme fragment complementation for the measurement of Wnt/β‐catenin signaling

5. Neurokinin-3 Receptor-Specific Antagonists Talnetant and Osanetant Show Distinct Mode of Action in Cellular Ca2+ Mobilization but Display Similar Binding Kinetics and Identical Mechanism of Binding in Ligand Cross-Competition

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