2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization-Reference-Cited by-同舟云学术

2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and Analogues as A2A Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization

Published:2005-10-01 Issue:22 Volume:48 Page:6887-6896
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Minetti Patrizia¹,Tinti Maria Ornella¹,Carminati Paolo¹,Castorina Massimo¹,Di Cesare Maria Assunta¹,Di Serio Stefano¹,Gallo Grazia¹,Ghirardi Orlando¹,Giorgi Fabrizio¹,Giorgi Luca¹,Piersanti Giovanni¹,Bartoccini Francesca¹,Tarzia Giorgio¹

Affiliation:

1. Istituto di Chimica Farmaceutica, Università degli Studi di Urbino “Carlo Bo”, Piazza del Rinascimento 6, 61029 Urbino (PU), and Italy, Dipartimento di Chimica and Dipartimento Sistema Nervoso Centrale e Periferico Sigma-Tau, via Pontina Km 30,400, 00040 Pomezia (Roma), Italy.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm058018d

Reference25 articles.

1. Adenosine receptors: new opportunities for future drugs

2. Adenosine A2A antagonists with potent anti-cataleptic activity

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