Synthesis and Biological Evaluation of Cyclopropyl Analogs of the Antiestrogen MER 25
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry
Reference31 articles.
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2. Synthesis and Biological Evaluation of gem- Dichlorocyclopropyl and Cyclopropyl Analogs of Stilbene Congeners as Potential Antiestrogens
3. Antiestrogens. 2. Structure-activity studies in a series of 3-aroyl-2-arylbenzo[b]thiophene derivatives leading to [6-hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl]-[4-[2-(1-piperidinyl)ethoxy]phenyl]methanone hydrochloride (LY 156758), a remarkably effective estrogen antagonist with only minimal intrinsic estrogenicity
4. 2-Phenylindoles. Relationship between structure, estrogen receptor affinity, and mammary tumor inhibiting activity in the rat
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1. Cytotoxic and Antimicrobial Activity of Dehydrozingerone based Cyclopropyl Derivatives;Chemistry & Biodiversity;2017-07-01
2. Design, synthesis, and biological evaluation of cyclopropyl analogues of stilbene with raloxifene side chain as subtype-selective ligands for estrogen receptor;Archives of Pharmacal Research;2013-04-24
3. Inhibition of Estrogen Receptor α-Mediated Transcription by Antiestrogenic 1,1-Dichloro-2,2,3-triarylcyclopropanes;Molecular Pharmacology;2004-07-02
4. N-Alkoxypyrazoles as biomimetics for the alkoxyphenyl group in tamoxifen;Bioorganic & Medicinal Chemistry;2003-04
5. Syntheses of gem-Dihalocyclopropanes and Their Use in Organic Synthesis;Chemical Reviews;2003-03-04
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