Design, synthesis, and biological evaluation of cyclopropyl analogues of stilbene with raloxifene side chain as subtype-selective ligands for estrogen receptor-Reference-Cited by-同舟云学术

Design, synthesis, and biological evaluation of cyclopropyl analogues of stilbene with raloxifene side chain as subtype-selective ligands for estrogen receptor

Published:2013-04-24 Issue:9 Volume:36 Page:1096-1103
ISSN:0253-6269
Container-title:Archives of Pharmacal Research
language:en
Short-container-title:Arch. Pharm. Res.

Author:

Yeo Hye Lim,Song Yoon Sun,Ryu Jae-Ha,Kim Hee-Doo

Publisher

Springer Science and Business Media LLC

Subject

Organic Chemistry,Drug Discovery,Molecular Medicine

Link

http://link.springer.com/content/pdf/10.1007/s12272-013-0134-2.pdf

Reference16 articles.

1. Ali, S., L. Buluwela, and R.C. Coombes. 2011. Antiestrogens and their therapeutic applications in breast cancer and other diseases. Annual Review of Medicine 62: 217–232.

2. Carpita, A., A. Ribecai, R. Rossi, and P. Stabile. 2002. Synthesis of the racemic forms of carbon–carbon double bond locked analogues of strobilurins which are characterized by a 2-arylcyclopropane ring cis-substituted at C-1 by the methyl (E)-3-methoxypropenoate unit. Tetrahedron 58: 3673–3680.

3. Catherino, W.H., and V.C. Jordan. 1995. Increasing the number of tandem estrogen response elements increases the estrogenic activity of a tamoxifen analogue. Cancer Letters 92: 39–47.

4. Chen, H.Y., K.D. Dykstra, E.T. Birzin, K. Frisch, W. Chan, Y.T. Yang, R.T. Mosley, F. DiNinno, S.P. Rohrer, J.M. Schaeffer, and M.L. Hammond. 2004. Estrogen receptor ligands. Part 1: The discovery of flavonoids with subtype selectivity. Bioorganic & Medicinal Chemistry Letters 14: 1417–1421.

5. Chlebowski, R.T., and G.L. Anderson. 2012. Changing concepts: Menopausal hormone therapy and breast cancer. Journal of the National Cancer Institute 104(7): 517–527.

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