A Series of 7-ω-carboxamidoalkyl-substituted estra-1,3,5(10),6-tetraenes-Reference-Cited by-同舟云学术

A Series of 7-ω-carboxamidoalkyl-substituted estra-1,3,5(10),6-tetraenes

Published:2002-01 Issue:1 Volume:2002 Page:1-3
ISSN:1747-5198
Container-title:Journal of Chemical Research
language:en
Short-container-title:Journal of Chemical Research

Author:

Thiemann Thies¹,Umeno Kuniharu²,Inohae Eiko²,Imai Masao²,Shima Yuji²,Mataka Shuntaro¹

Affiliation:

1. Institute of Advanced Material Study, 6-1, Kasuga-koh-en, Kasuga-shi, Fukuoka 816-8580, Japan

2. Graduate School of Engineering, Kyushu University, 6-1, Kasuga-koh-en, Kasuga-shi, Fukuoka 816-8580, Japan

Abstract

A number of 7-ω-carboxamidoalkyl-substituted estra-1,3,5(10),6-tetraenes as potential ligands for the estrogen receptor ERα have been prepared using either a conjugate addition of α,ω-iodoalkanenitriles or a Michael addition to steroidal ketone 3 as the key step.

Publisher

SAGE Publications

Subject

General Chemistry

Link

http://journals.sagepub.com/doi/pdf/10.3184/030823402103170312

Reference7 articles.

1. Comparative QSAR Analysis of Estrogen Receptor Ligands

2. Synthesis and biological evaluation of two new radiolabelled estrogens: [125I](E)-3-methoxy-17α-iodovinylestra-1,3,5(10),6-tetraen-17β-ol and [125I](Z)-3-methoxy-17α-iodovinylestra-1,3,5(10),6-tetraen-17β-ol

3. AN EXPEDITIOUS ROUTE TO 7α-SUBSTITUTED ESTRADIOL DERIVATIVES

4. A stereoselective synthesis of 7α-(3′-carboxypropyl)estradiol from a noncontrolled substance

5. Synthesis and estrogenic activities of novel 7-thiosubstituted estratriene derivatives

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