Efficient Synthesis of Substituted 2-(4H-1,3-benzoxazin-2-yl)Phenols via a Pseudo Three-Component Reaction-Reference-Cited by-同舟云学术

Efficient Synthesis of Substituted 2-(4H-1,3-benzoxazin-2-yl)Phenols via a Pseudo Three-Component Reaction

Published:2018-03 Issue:3 Volume:42 Page:121-124
ISSN:1747-5198
Container-title:Journal of Chemical Research
language:en
Short-container-title:Journal of Chemical Research

Author:

Wang Ting¹,Dai Chenlu¹,Qing Xushun¹,Wang Cunde

Affiliation:

1. School of Chemistry and Chemical Engineering, Yangzhou University, 180 Siwangting Street, Yangzhou 225002, P.R. China

Abstract

An efficient pseudo three-component reaction between substituted 2-hydroxybenzaldehydes and ammonium acetate for the preparation of substituted 2-(4 H-1,3-benzoxazin-2-yl)phenols in moderate to good yields (70-80%) was developed. The structure of a typical product was confirmed by X-ray crystallography.

Publisher

SAGE Publications

Subject

General Chemistry

Link

http://journals.sagepub.com/doi/pdf/10.3184/174751918X15199181776822

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