Structurally Related Kappa Opioid Receptor Agonists with Substantial Differential Signaling Bias: Neuroendocrine and Behavioral Effects in C57BL6 Mice
Author:
Affiliation:
1. Laboratory of the Biology of Addictive Diseases, Rockefeller University, New York, New York
Funder
Robertson Therapeutic Development Fund
Dr. Miriam and Sheldon G. Adelson Medical Research Foundation
Publisher
Oxford University Press (OUP)
Subject
Pharmacology (medical),Psychiatry and Mental health,Pharmacology
Link
http://academic.oup.com/ijnp/article-pdf/21/9/847/25645736/pyy034.pdf
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3. Differential effects of the novel kappa opioid receptor antagonist, jdtic, on reinstatement of cocaine-seeking induced by footshock stressors vs cocaine primes and its antidepressant-like effects in rats;Beardsley;Psychopharmacology (Berl),2005
4. Operational models of pharmacological agonism;Black;Proc R Soc Lond B Biol Sci,1983
5. Approaches to assess functional selectivity in gpcrs: evaluating G protein signaling in an endogenous environment;Bohn;Methods Mol Biol,2015
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