Inhibition of poly(ADP‐ribose) polymerase prevents irinotecan‐induced intestinal damage and enhances irinotecan/temozolomide efficacy against colon carcinoma

Author:

Tentori Lucio1,Leonetti Carlo2,Scarsella Marco2,Muzi Alessia1,Mazzon Emanuela3,Vergati Matteo1,Forini Olindo1,Lapidus Rena4,Xu Weizheng4,Dorio Annalisa Susanna1,Zhang Jie4,Cuzzocrea Salvatore3,Graziani Grazia1,Tentori Lucio1,Leonetti Carlo2,Scarsella Marco2,Muzi Alessia1,Mazzon Emanuela3,Vergati Matteo1,Forini Olindo1,Lapidus Rena4,Xu Weizheng4,Dorio Annalisa Susanna1,Zhang Jie4,Cuzzocrea Salvatore3,Grazia Grazia1

Affiliation:

1. Department of NeuroscienceUniversity of Rome “Tor Vergata,”RomeItaly

2. Experimental Clinical LaboratoryInstitute for Cancer Research “Regina Elena,”RomeItaly

3. Department of Clinical and Experimental Medicine and PharmacologyUniversity of Messina“Centro Neurolesi Bonino-Pulejo” (IRCCS)MessinaItaly

4. MGI PharmaBaltimoreMarylandUSA

Publisher

Wiley

Subject

Genetics,Molecular Biology,Biochemistry,Biotechnology

Reference48 articles.

1. Irinotecan combined with fluorouracil compared with fluorouracil alone as first-line treatment for metastatic colorectal cancer: a multicentre randomised trial

2. Mechanisms of resistance to topoisomerase I-targeting drugs

3. Antitumor activity of temozolomide combined with irinotecan is partly independent of O6-methylguanine-DNA methyltransferase and mismatch repair phenotypes in xenograft models;Houghton P. J.;Clin. Cancer Res.,2000

4. Schedule-dependent activity of temozolomide plus CPT-11 against a human central nervous system tumor-derived xenograft;Patel V. J.;Clin. Cancer Res.,2000

5. Trial of irinotecan and temozolomide in patients with solid tumors;Jones S. F.;Oncology,2003

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