Development of a High-Throughput Screen to Detect Inhibitors of TRPS1 Sumoylation
Author:
Affiliation:
1. Molecular Discovery Research, GlaxoSmithKline, Collegeville, Pennsylvania.
Publisher
Mary Ann Liebert Inc
Subject
Drug Discovery,Molecular Medicine
Link
http://www.liebertpub.com/doi/pdf/10.1089/adt.2012.501
Reference41 articles.
1. Protein Modification by SUMO
2. The SUMO pathway: emerging mechanisms that shape specificity, conjugation and recognition
3. Structural Basis for E2-Mediated SUMO Conjugation Revealed by a Complex between Ubiquitin-Conjugating Enzyme Ubc9 and RanGAP1
4. Identification of a Substrate Recognition Site on Ubc9
5. The Small Ubiquitin-like Modifier-1 (SUMO-1) Consensus Sequence Mediates Ubc9 Binding and Is Essential for SUMO-1 Modification
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