The Cellular Distribution of Fluorescently Labeled Arrestins Provides a Robust, Sensitive, and Universal Assay for Screening G Protein-Coupled Receptors-Reference-Cited by-同舟云学术

The Cellular Distribution of Fluorescently Labeled Arrestins Provides a Robust, Sensitive, and Universal Assay for Screening G Protein-Coupled Receptors

Published:2002-11 Issue:1 Volume:1 Page:21-30
ISSN:1540-658X
Container-title:ASSAY and Drug Development Technologies
language:en
Short-container-title:ASSAY and Drug Development Technologies

Author:

Oakley Robert H.¹,Hudson Christine C.²,Cruickshank Rachael D.²,Meyers Diane M.²,Payne Richard E.²,Rhem Shay M.²,Loomis Carson R.²

Affiliation:

1. Norak Biosciences, Inc., Research Triangle Park, NC.

2. Biosciences, Inc., Research Triangle Park, NC.

Publisher

Mary Ann Liebert Inc

Subject

Drug Discovery,Molecular Medicine

Link

http://www.liebertpub.com/doi/pdf/10.1089/154065802761001275

Reference40 articles.

1. Patent status of the therapeutically important G-protein-coupled receptors

2. THE ROLE OF RECEPTOR KINASES AND ARRESTINS IN G PROTEIN–COUPLED RECEPTOR REGULATION

3. A β-Arrestin/Green Fluorescent Protein Biosensor for Detecting G Protein-coupled Receptor Activation

4. Receptor-specific desensitization with purified proteins. Kinase dependence and receptor specificity of beta-arrestin and arrestin in the beta 2-adrenergic receptor and rhodopsin systems.

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