Structural determinants influencing halogen bonding: a case study on azinesulfonamide analogs of aripiprazole as 5-HT1A, 5-HT7, and D2 receptor ligands-Reference-Cited by-同舟云学术

Structural determinants influencing halogen bonding: a case study on azinesulfonamide analogs of aripiprazole as 5-HT1A, 5-HT7, and D2 receptor ligands

Published:2018-05-11 Issue:1 Volume:12 Page:
ISSN:1752-153X
Container-title:Chemistry Central Journal
language:en
Short-container-title:Chemistry Central Journal

Author:

Marciniec Krzysztof^ORCID,Kurczab Rafał,Książek Maria,Bębenek Ewa,Chrobak Elwira,Satała Grzegorz,Bojarski Andrzej J.,Kusz Joachim,Zajdel Paweł

Publisher

Springer Science and Business Media LLC

Subject

General Chemistry

Link

http://link.springer.com/content/pdf/10.1186/s13065-018-0422-5.pdf

Reference47 articles.

1. Volk B, Gacsalyi I, Pallagi K, Poszawacz L, Gyonos I, Szabo E, Bako T, Spedding M, Simig G, Szenasi G (2011) Optimization of (arylpiperazinylbutyl)oxindoles exhibiting selective 5-HT7 receptor antagonist activity. J Med Chem 54:6657–6669

2. Butini S, Gemma S, Campiani G, Franceschini S, Trotta F, Borriello M, Ceres N, Ros S, Sanna Coccone S, Bernetti M, De Angelis M, Brindisi M, Nacci V, Fiorini I, Novellino E, Cagnotto A, Mennini T, Sandager-Nielsen K, Andreasen JT, Scheel-Kruger J, Mikkelsen JD, Fattorusso C (2009) Discovery of a new class of potential multifunctional atypical antipsychotic agents targeting dopamine D3 and serotonin 5-HT1A and 5-HT2A receptors: design, synthesis, and effects on behavior. J Med Chem 52:151–169

3. Leopoldo M, Berardi F, Colabufo NA, De Giorgio P, Lacivita E, Perrone R, Tortorella V (2002) Structure–affinity relationship study on N-[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D3 receptor ligands. J Med Chem 45:5727–5735

4. Zajdel P, Partyka A, Marciniec K, Bojarski AJ, Pawłowski M, Wesołowska A (2014) Quinoline- and isoquinoline-sulfonamide analogs of aripiprazole: novel antipsychotic agents? Future Med Chem 6:1–19

5. Zajdel P, Marciniec K, Maślankiewicz A, Grychowska K, Satała G, Duszyńska B, Lenda T, Siwek A, Nowak G, Partyka A, Wróbel D, Jastrzębska-Więsek M, Bojarski AJ, Wesołowska A, Pawłowski M (2013) Antidepressant and antipsychotic activity of new quinoline- and isoquinoline-sulfonamide analogs of aripiprazole targeting serotonin 5-HT1A/5-HT2A/5-HT7 and dopamine D2/D3 receptors. Eur J Med Chem 60:42–50

Cited by 8 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Halogen Bonding Hot Spots as a Constraint in Virtual Screening: A Case Study of 5-HT₇R;Journal of Medicinal Chemistry;2024-07-31

2. Development and challenges in the discovery of 5-HT1A and 5-HT7 receptor ligands;Bioorganic Chemistry;2023-02

3. Recent Advances in Biological Active Sulfonamide-based Hybrid Compounds Part C: Multicomponent Sulfonamide Hybrids;Current Medicinal Chemistry;2022-11-28

4. A new class of 5-HT1A receptor antagonists with procognitive and antidepressant properties;Future Medicinal Chemistry;2021-09

5. Chlorine substituents and linker topology as factors of 5-HT6R activity for novel highly active 1,3,5-triazine derivatives with procognitive properties in vivo;European Journal of Medicinal Chemistry;2020-10