Synthesis, biological evaluation and molecular docking studies of 6-(4-nitrophenoxy)-1H-imidazo[4,5-b]pyridine derivatives as novel antitubercular agents: future DprE1 inhibitors
Author:
Publisher
Springer Science and Business Media LLC
Subject
General Chemistry
Link
http://link.springer.com/content/pdf/10.1186/s13065-018-0515-1.pdf
Reference50 articles.
1. Batt SM, Jabeen T, Bhowruth V, Quill L, Lund PA, Eggeling L (2012) Structural basis of inhibition of Mycobacterium tuberculosis DprE1 by benzothiazinones inhibitors. Proc Natl Acad Sci 109:354–359. https://doi.org/10.1073/pnas.1205735109
2. Riccardi G, Pasca MR, Chiarelli LR, Manina G, Mattevi A, Binda C (2013) The DprE1 enzyme, one of the most vulnerable targets of Mycobacterium tuberculosis. Appl Microbiol Biotechnol 97:8841–8848. https://doi.org/10.1007/s00253-013-5218-x
3. Makarov V, Neres J, Hartkoorn RC, Ryabova OB, Kazakova E, Šarkan M (2015) 8-Pyrrole-benzothiazinones non-covalent inhibitors of DprE1 from Mycobacterium tuberculosis. Antimicrob Agents Chemother 59:778–786. https://doi.org/10.1128/AAC.00778-15
4. Scribner A, Dennis R, Lee S, Ouvry G, Perrey D, Fisher M (2008) Synthesis and biological activity of imidazopyridine anticoccidial agents: part II. Eur J Med Chem 43:1123–1151. https://doi.org/10.1016/j.ejmech.2007.02.006
5. Piton J, Foo CSY, Cole ST (2017) Structural studies of Mycobacterium tuberculosis DprE1 interacting with its inhibitors. Drug discov today 22:526–533. https://doi.org/10.1016/j.drudis.2016.09.014
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