Beta-Blockers Show Inverse Agonism to a Novel Constitutively Active Mutant of β1-Adrenoceptor-Reference-Cited by-同舟云学术

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Beta-Blockers Show Inverse Agonism to a Novel Constitutively Active Mutant of β1-Adrenoceptor

Published:2006 Issue:2 Volume:102 Page:167-172
ISSN:1347-8613
Container-title:Journal of Pharmacological Sciences
language:en
Short-container-title:J Pharmacol Sci

Author:

Ahmed Maruf,Muntasir Habib Abul,Hossain Murad,Ishiguro Masaji,Komiyama Tadazumi,Muramatsu Ikunobu,Kurose Hitoshi,Nagatomo Takafumi

Publisher

Japanese Pharmacological Society

Subject

Pharmacology,Molecular Medicine

Reference28 articles.

1. 1 Weiss J. G-protein-coupled receptors: molecular mechanisms involved in receptor activation and selectivity of G-protein recognition. FASEB J. 1997;5:346–354.

2. Constitutive activity of G-protein-coupled receptors: cause of disease and common property of wild-type receptors

3. Regions of the alpha 1-adrenergic receptor involved in coupling to phosphatidylinositol hydrolysis and enhanced sensitivity of biological function.

4. 4 Kjelsberg MA, Cotecchia S, Ostrowski J, Caron MG, Lefkowitz RJ. Constitutive activation of the α_1B-adrenergic receptor by all amino acid substitution at a single site. J Biol Chem. 1992;67:1430–1433.

5. 5 Ren Q, Kurose H, Lefkowitz RJ, Cotecchia S. Constitutively active mutants of the α_2A-adrenergic receptor. J Biol Chem. 1993;68:16483–16487.

Cited by 8 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Insights into the Role of Asp792.50 in β2 Adrenergic Receptor Activation from Molecular Dynamics Simulations;Biochemistry;2014-11-12

2. The 2.1 Å Resolution Structure of Cyanopindolol-Bound β1-Adrenoceptor Identifies an Intramembrane Na+ Ion that Stabilises the Ligand-Free Receptor;PLoS ONE;2014-03-24

3. A Conserved Protonation-Induced Switch can Trigger “Ionic-Lock” Formation in Adrenergic Receptors;Journal of Molecular Biology;2010-04

4. MEASUREMENT OF INVERSE AGONISM IN beta-ADRENOCEPTORS;METHOD ENZYMOL;2010

5. Measurement of Inverse Agonism in β-Adrenoceptors;Methods in Enzymology;2010

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