Synthesis of Azole Derivatives of 1,2,3-Dithiazole-5-imines and Study of Their Fungicidal

Author:

Tsaplin G. V.ORCID,Bashkalova E. I.,Alekseenko A. L.ORCID,Popkov S. V.ORCID

Abstract

Abstract A three-stage method was proposed for the synthesis of new 4-[4-(2-azolylethyl)piperazine-1-yl]-N-aryl-5H-1,2,3-dithiazole-5-imines. This approach includes the reaction of Appel salt with anilines to produce 1,2,3-dithiazole-5-imines, which were converted into 4-[(4-chloroethyl)piperazine-1-yl]-5H-1,2,3-dithiazole-5-imines, alkylating azoles at the final stage. The high fungicidal activity of target compounds and intermediate 4-chloro-N-aryl-1,2,3-dithiazole-5-imines was shown in vitro tests versus six species of phytopathogenic fungi.

Publisher

Pleiades Publishing Ltd

Subject

General Chemistry

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