Effect of Usnic Acid-Derived Tyrosyl-DNA Phosphodiesterase 1 Inhibitor Used as Monotherapy or in Combination with Olaparib on Transplanted Tumors In Vivo

Author:

Kornienko T. E.,Zakharenko A. L.,Ilina E. S.,Chepanova A. A.,Zakharova O. D.,Dyrkheeva N. S.,Popova N. A.,Nikolin V. P.,Filimonov A. S.,Luzina O. A.,Salakhutdinov N. F.,Lavrik O. I.

Publisher

Pleiades Publishing Ltd

Subject

Structural Biology,Biophysics

Reference21 articles.

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2. Curtin N.J., Szabo C. 2020. Poly (ADP-ribose) polymerase inhibition: past, present and future. Nat. Rev. Drug Discov. 19, 711–736.

3. Zakharenko A., Dyrkheeva N., Lavrik O. 2019. Dual DNA topoisomerase 1 and tyrosyl-DNA phosphodiesterase 1 inhibition for improved anticancer activity. Med. Res. Rev. 39, 1427–1441.

4. Alagoz M., Gilbert D.C., El-Khamisy S., Chalmers A.J. 2012. DNA repair and resistance to topoisomerase I inhibitors: mechanisms, biomarkers and therapeutic targets. Curr. Med. Chem. 19, 3874–3885.

5. Pommier Y., Huang S.N., Gao R., Das B.B., Murai J., Marchand C. 2014. Tyrosyl-DNA-phosphodiesterases (tdp1 and tdp2). DNA Repair. 19, 114–129.

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