Interspecies scaling of tolcapone, a new inhibitor of catechol-O-methyltransferase (COMT). Use ofin vitrodata from hepatocytes to predict metabolic clearance in animals and humans-Reference-Cited by-同舟云学术

Interspecies scaling of tolcapone, a new inhibitor of catechol-O-methyltransferase (COMT). Use ofin vitrodata from hepatocytes to predict metabolic clearance in animals and humans

Published:1996-01 Issue:8 Volume:26 Page:839-851
ISSN:0049-8254
Container-title:Xenobiotica
language:en
Short-container-title:Xenobiotica

Author:

Lave Th.,Dupin S.,Schmitt M.,Kapps M.,Meyer J.,Morgenroth B.,Chou R. C.,Jaeck D.,Coassolo Ph.

Publisher

Informa UK Limited

Subject

Health, Toxicology and Mutagenesis,Pharmacology,Toxicology,Biochemistry,General Medicine

Link

http://www.tandfonline.com/doi/pdf/10.3109/00498259609046754

Reference21 articles.

1. Scaling of antipyrine intrinsic clearance of unbound drug in 15 mammalian species

2. Animal phannacokinetics and interspecies scaling of FCE 22101, a penem antibiotic

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