Utility of the carboxylesterase inhibitorbis-para-nitrophenylphosphate (BNPP) in the plasma unbound fraction determination for a hydrolytically unstable amide derivative and agonist of the TGR5 receptor-Reference-Cited by-同舟云学术

Utility of the carboxylesterase inhibitorbis-para-nitrophenylphosphate (BNPP) in the plasma unbound fraction determination for a hydrolytically unstable amide derivative and agonist of the TGR5 receptor

Published:2010-03-18 Issue:6 Volume:40 Page:369-380
ISSN:0049-8254
Container-title:Xenobiotica
language:en
Short-container-title:Xenobiotica

Author:

Eng H.,Niosi M.,McDonald T. S.,Wolford A.,Chen Y.,Simila S. T. M.,Bauman J. N.,Warmus J.,Kalgutkar A. S.

Publisher

Informa UK Limited

Subject

Health, Toxicology and Mutagenesis,Pharmacology,Toxicology,Biochemistry,General Medicine

Link

http://www.tandfonline.com/doi/pdf/10.3109/00498251003706598

Reference56 articles.

1. Stereospecific activity and nature of metabolizing esterases for propranolol prodrug in hairless mouse skin, liver and plasma

2. GLP-1 based therapy for type 2 diabetes

3. MULTIPLE FORMS OF ESTERASE IN VERTEBRATE BLOOD PLASMA*

4. EFFECTIVE DOSING REGIMEN OF 1-AMINOBENZOTRIAZOLE FOR INHIBITION OF ANTIPYRINE CLEARANCE IN GUINEA PIGS AND MICE USING SERIAL SAMPLING

Cited by 51 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Pharmacokinetics of Panobinostat: Interspecies Difference in Metabolic Stability;Journal of Pharmacology and Experimental Therapeutics;2024-02-26

2. Distribution - In Vitro Test: Protein Binding;Drug Discovery and Evaluation: Safety and Pharmacokinetic Assays;2024

3. Biotransformation and brain distribution of the anti-COVID-19 drug molnupiravir and herb-drug pharmacokinetic interactions between the herbal extract Scutellaria formula-NRICM101;Journal of Pharmaceutical and Biomedical Analysis;2023-09

4. Alcohol inhibits the metabolism of dimethyl fumarate to the active metabolite responsible for decreasing relapse frequency in the treatment of multiple sclerosis;PLOS ONE;2022-11-28

5. Mouse Pharmacokinetics and In Vitro Metabolism of SH-11037 and SH-11008, Synthetic Homoisoflavonoids for Retinal Neovascularization;Pharmaceutics;2022-10-24