A squaramide-catalysed asymmetric cascade Michael addition/acyl transfer reaction between unsaturated benzothiophenones and α-nitroketones-Reference-Cited by-同舟云学术

A squaramide-catalysed asymmetric cascade Michael addition/acyl transfer reaction between unsaturated benzothiophenones and α-nitroketones

Published:2022 Issue:4 Volume:20 Page:840-846
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Niu Cheng¹,Du Da-Ming¹^ORCID

Affiliation:

1. Key Laboratory of Medical Molecule Science & Pharmaceutics Engineering, Ministry of Industry and Information Technology, School of Chemistry and Chemical Engineering, Beijing Institute of Technology, No. 5 Zhongguancun South Street, Beijing 100081, People's Republic of China

Abstract

A practical organocatalytic asymmetric synthesis of chiral acyloxybenzothiophene derivatives was developed using unsaturated benzothiophenones and α-nitroketones catalysed by squaramide via Michael addition/acyl transfer cascade reactions.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2022/OB/D1OB02217B

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