Rhodium(iii)-catalyzed synthesis of 3-trifluoromethylindanones from N-methoxybenzamides via C–H activation and Claisen/retro-Claisen reaction-Reference-Cited by-同舟云学术

Rhodium(iii)-catalyzed synthesis of 3-trifluoromethylindanones from N-methoxybenzamides via C–H activation and Claisen/retro-Claisen reaction

Published:2020 Issue:12 Volume:7 Page:1512-1519
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Chaudhary Bharatkumar¹²³⁴⁵^ORCID,Kulkarni Neeraj¹²³⁴⁵^ORCID,Sharma Satyasheel¹²³⁴⁵^ORCID

Affiliation:

1. Department of Medicinal Chemistry

2. National Institute of Pharmaceutical Education and Research

3. Ahmedabad (NIPER-A)

4. Gandhinagar

5. India

Abstract

An efficient synthesis of 3-trifluoromethylindanones via C–H annulation of N-methoxybenzamides with β-trifluoromethyl-α,β-unsaturated ketones under Rh(iii)-catalysis is described.

Funder

Department of Science and Technology, Ministry of Science and Technology, India

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/QO/D0QO00330A

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