Catalytic enantioselective hydrophosphinylation of <i>in situ</i>-generated indole-derived vinylogous imines to access 3-(1-diphenylphosphoryl-arylmethyl)indoles-Reference-Cited by-同舟云学术

Catalytic enantioselective hydrophosphinylation of in situ-generated indole-derived vinylogous imines to access 3-(1-diphenylphosphoryl-arylmethyl)indoles

Published:2022 Issue:86 Volume:58 Page:12062-12065
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Jia Yun-Qing¹²³,Zhao Jian-Qiang²^ORCID,Wang Zhen-Hua²^ORCID,You Yong²^ORCID,Zhang Yan-Ping²,Jin Xin⁴,Zhou Ming-Qiang¹³,Ge Zhen-Zhen¹³,Yuan Wei-Cheng¹²^ORCID

Affiliation:

1. National Engineering Research Center of Chiral Drugs, Chengdu Institute of Organic Chemistry, Chinese Academy of Sciences, Chengdu, 610041, China

2. Innovation Research Center of Chiral Drugs, Institute for Advanced Study, Chengdu University, Chengdu, 610106, China

3. University of Chinese Academy of Sciences, Beijing, 100049, China

4. Zhejiang Jinhua Conba Bio-Pharm. Co. Ltd, Jinhua, 321016, China

Abstract

An efficient organocatalyzed enantioselective hydrophosphinylation of indole-derived vinylogous imines generated in situ from sulfonyl indoles was developed for the synthesis of optically active 3-(1-diphenylphosphoryl-arylmethyl)indoles.

Funder

National Natural Science Foundation of China

Sichuan Province Science and Technology Support Program

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2022/CC/D2CC04763B

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