Pd-Catalyzed direct C–H arylation of pyrrolo[1,2-a]quinoxalines-Reference-Cited by-同舟云学术

Pd-Catalyzed direct C–H arylation of pyrrolo[1,2-a]quinoxalines

Published:2022 Issue:4 Volume:20 Page:847-851
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Hao Di¹,Yang Zhen¹,Liu Yali¹,Li Yang¹,Li Chuntian¹,Gu Yanlong²^ORCID,Vaccaro Luigi³^ORCID,Liu Jichang¹,Liu Ping¹^ORCID

Affiliation:

1. School of Chemistry and Chemical Engineering, the Key Laboratory for Green Processing of Chemical Engineering of Xinjiang Bingtuan, Shihezi University, Shihezi City, 832004, China

2. Key Laboratory of Material Chemistry for Energy Conversion and Storage, Ministry of Education, Hubei Key Laboratory of Material Chemistry and Service Failure, School of Chemistry and Chemical Engineering, Huazhong University of Science & Technology, Wuhan City, 430074, China

3. Laboratory of Green S.O.C., Dipartimento di Chimica, Biologia e Biotecnologie, Università degli Studi di Perugia, Perugia, Italy

Abstract

An efficient Pd-catalyzed direct C–H arylation of pyrrolo[1,2-a]quinoxalines with aryl iodides is described, providing a series of 1-arylated and 1,3-diarylated pyrrolo[1,2-a]quinoxalines in good yields.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2022/OB/D1OB02248B

Reference46 articles.

1. Recent Progress in Biological Activities and Synthetic Methodologies of Pyrroloquinoxalines

2. Quinoxalinylethylpyridylthioureas (QXPTs) as Potent Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further SAR Studies and Identification of a Novel Orally Bioavailable Hydrazine-Based Antiviral Agent

3. Arylguanidine and arylbiguanide binding at 5-HT3 serotonin receptors: A QSAR study