A shortcut to high-affinity Ga-68 and Cu-64 radiopharmaceuticals: one-pot click chemistry trimerisation on the TRAP platform-Reference-Cited by-同舟云学术

A shortcut to high-affinity Ga-68 and Cu-64 radiopharmaceuticals: one-pot click chemistry trimerisation on the TRAP platform

Published:2015 Issue:24 Volume:44 Page:11137-11146
ISSN:1477-9226
Container-title:Dalton Transactions
language:en
Short-container-title:Dalton Trans.

Author:

Baranyai Zsolt¹²³⁴,Reich Dominik⁵⁶⁷⁸,Vágner Adrienn¹²³⁴,Weineisen Martina⁵⁶⁷⁸,Tóth Imre¹²³⁴,Wester Hans-Jürgen⁵⁶⁷⁸,Notni Johannes⁵⁶⁷⁸

Affiliation:

1. Department of Inorganic and Analytical Chemistry

2. University of Debrecen

3. Debrecen

4. Hungary

5. Lehrstuhl für Pharmazeutische Radiochemie

6. Technische Universität München

7. D-85748 Garching

8. Germany

Abstract

The kinetic inertness profile of Cu(ii) complexes of TRAP-conjugates enables simple Cu(ii) removal after click functionalisation and confirms their suitability for Cu-64-PET.

Funder

Deutsche Forschungsgemeinschaft

Országos Tudományos Kutatási Alapprogramok

Publisher

Royal Society of Chemistry (RSC)

Subject

Inorganic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2015/DT/C5DT00576K

Reference76 articles.

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