Converting oxazoles into imidazoles: new opportunities for diversity-oriented synthesis-Reference-Cited by-同舟云学术

Converting oxazoles into imidazoles: new opportunities for diversity-oriented synthesis

Published:2014 Issue:15 Volume:50 Page:1867-1870
ISSN:1359-7345
Container-title:Chem. Commun.
language:en
Short-container-title:Chem. Commun.

Author:

Alzieu Thibaut¹²³⁴⁵,Lehmann Johannes¹²³⁴⁵,Naidu Ajay B.⁶⁷⁸,Martin Rainer E.¹²³⁴⁵,Britton Robert⁶⁷⁸

Affiliation:

1. Medicinal Chemistry

2. Small Molecule Research

3. Pharma Research & Early Development (pRED)

4. F. Hoffmann-La Roche AG

5. 4070 Basel, Switzerland

6. Department of Chemistry

7. Simon Fraser University

8. Burnaby, Canada

Abstract

We report the optimization of a neglected reaction for the rapid and direct conversion of oxazoles into N-substituted imidazoles.

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2014/CC/C3CC48467J

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