Late stage iodination of biologically active agents using a one-pot process from aryl amines-Reference-Cited by-同舟云学术

Late stage iodination of biologically active agents using a one-pot process from aryl amines

Published:2017 Issue:86 Volume:7 Page:54881-54891
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Sloan Nikki L.¹²³⁴⁵,Luthra Sajinder K.⁶⁷⁸⁹,McRobbie Graeme⁶⁷⁸⁹,Pimlott Sally L.¹⁰¹¹¹²⁹,Sutherland Andrew¹²³⁴⁵^ORCID

Affiliation:

1. WestCHEM

2. School of Chemistry

3. The Joseph Black Building

4. University of Glasgow

5. Glasgow G12 8QQ

6. GE Healthcare

7. The Grove Centre

8. Amersham

9. UK

10. West of Scotland PET Centre

11. Greater Glasgow and Clyde NHS Trust

12. Glasgow G12 0YN

Abstract

A tandem process has been developed for the general preparation of aryl iodide compounds from anilines that is also applicable for the late-stage iodination of biologically active agents.

Funder

Medical Research Scotland

GE Healthcare

University of Glasgow

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/RA/C7RA11860K

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