Facile synthesis of chiral ε-sultams via an organocatalytic aza-Friedel–Crafts reaction-Reference-Cited by-同舟云学术

Facile synthesis of chiral ε-sultams via an organocatalytic aza-Friedel–Crafts reaction

Published:2019 Issue:26 Volume:17 Page:6364-6368
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Zhao Zi-Biao¹²³⁴⁵^ORCID,Shi Lei¹²³⁴⁵^ORCID,Li Yaming¹²³⁴⁵,Meng Fan-Jie¹²³⁴⁵,Zhou Yong-Gui¹²³⁴⁵^ORCID

Affiliation:

1. State Key Laboratory of Fine Chemicals

2. Zhang Dayu School of Chemistry

3. Dalian University of Technology

4. Dalian 116024

5. P. R. China

Abstract

A facile enantioselective aza-Friedel–Crafts reaction has been developed for the synthesis of chiral ε-sultams with an enantiomeric excess of up to 92%.

Funder

National Natural Science Foundation of China

Dalian Science and Technology Bureau

Chinese Academy of Sciences

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2019/OB/C9OB01158G

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