Transition-metal-free oxidative C5 C–H-halogenation of 8-aminoquinoline amides using sodium halides-Reference-Cited by-同舟云学术

Transition-metal-free oxidative C5 C–H-halogenation of 8-aminoquinoline amides using sodium halides

Published:2016 Issue:43 Volume:14 Page:10180-10184
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Wang Ying¹²³⁴,Wang Yang¹²³⁴,Jiang Kai¹²³⁴,Zhang Qian¹²³⁴⁵,Li Dong¹²³⁴^ORCID

Affiliation:

1. School of Materials and Chemical Engineering

2. Hubei University of Technology

3. Wuhan 430068

4. China

5. Hubei Key Laboratory of Drug Synthesis and Optimization

Abstract

A simple and efficient transition-metal-free oxidative halogenation (Cl, Br) of the C5 C–H bond of 8-aminoquinoline amides, with low-cost and innoxious sodium halides, has been developed.

Funder

National Natural Science Foundation of China

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/OB/C6OB02079H

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