Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity-Reference-Cited by-同舟云学术

Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity

Published:2024 Issue:6 Volume:15 Page:1929-1941
ISSN:2632-8682
Container-title:RSC Medicinal Chemistry
language:en
Short-container-title:RSC Med. Chem.

Author:

Aslan Hakan¹²^ORCID,Renzi Gioele²,Angeli Andrea²^ORCID,D'Agostino Ilaria²³^ORCID,Ronca Roberto⁴^ORCID,Massardi Maria Luisa⁴^ORCID,Tavani Camilla⁴^ORCID,Carradori Simone⁵^ORCID,Ferraroni Marta⁶^ORCID,Governa Paolo⁷^ORCID,Manetti Fabrizio⁷^ORCID,Carta Fabrizio²^ORCID,Supuran Claudiu T.²^ORCID

Affiliation:

1. Department of Chemistry, Faculty of Science and Arts, Sinop University, Sinop, Turkey

2. NEUROFARBA Department, Sezione di Scienze Farmaceutiche, University of Florence, Sesto Fiorentino, Florence, 50019, Italy

3. Department of Pharmacy, University of Pisa, 56126, Pisa, Italy

4. Department of Molecular and Translational Medicine, University of Brescia, 25123 Brescia, Italy

5. Department of Pharmacy, “G. d'Annunzio” University of Chieti-Pescara, 66100 Chieti, Italy

6. Department of Chemistry “Ugo Schiff”, University of Florence, Sesto Fiorentino, Florence, 50019, Italy

7. Department of Biotechnology, Chemistry and Pharmacy, University of Siena, 53100, Siena, Italy

Abstract

One-step synthesis and a chemical similarity-based screening provide new tumor-associated carbonic anhydrase (CA) inhibitors for anticancer application.

Funder

Scientific and Technological Research Council of Turkey

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/MD/D4MD00101J

Reference61 articles.

1. Cancer statistics, 2023

2. Word Health Organization. Cancer [Internet], [cited 2023 Sep 13], Available from: https://www.who.int/news-room/fact-sheets/detail/cancer

3. The Burden of Illness of Cancer: Economic Cost and Quality of Life

4. CRISPR applications in cancer diagnosis and treatment

5. Ten Years of CRISPRing Cancers In Vitro

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