Synthesis of substituted 3,4-dihydroquinazolinones via a metal free Leuckart–Wallach type reaction-Reference-Cited by-同舟云学术

Synthesis of substituted 3,4-dihydroquinazolinones via a metal free Leuckart–Wallach type reaction

Published:2021 Issue:1 Volume:11 Page:349-353
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Bokale-Shivale Suvarna¹²³⁴⁵,Amin Mohammad A.¹²³⁴⁵^ORCID,Sawant Rajiv T.¹²³⁴⁵,Stevens Marc Y.¹²³⁴⁵,Turanli Lewend¹²³⁴⁵,Hallberg Adam¹²³⁴⁵,Waghmode Suresh B.⁶⁷⁸⁹^ORCID,Odell Luke R.¹²³⁴⁵^ORCID

Affiliation:

1. Department of Medicinal Chemistry

2. Uppsala Biomedical Center

3. Uppsala University

4. SE-751 23 Uppsala

5. Sweden

6. Department of Chemistry

7. Savitribai Phule Pune University (formerly Pune University)

8. Pune 411 007

9. India

Abstract

A novel cascade cyclization/Leuckart–Wallach type strategy to prepare biologically important 3,4-dihydroquinazolinones is presented.

Funder

Vetenskapsrådet

Uppsala Universitet

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2021/RA/D0RA10142G

Reference42 articles.

1. Calcitonin Gene-Related Peptide Receptor Antagonists: New Therapeutic Agents for Migraine

2. Inhibition of Clinically Relevant Mutant Variants of HIV-1 by Quinazolinone Non-Nucleoside Reverse Transcriptase Inhibitors

3. Discovery of dihydroquinazolinone derivatives as potent, selective, and CNS-penetrant M1 and M4 muscarinic acetylcholine receptors agonists

4. Quinazolinone-Based Anticancer Agents: Synthesis, Antiproliferative SAR, Antitubulin Activity, and Tubulin Co-crystal Structure

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