Copper-catalyzed synthesis of aminoquinolines from β-(2-aminophenyl)-α,β-ynones using DMF as dual synthon-Reference-Cited by-同舟云学术

Copper-catalyzed synthesis of aminoquinolines from β-(2-aminophenyl)-α,β-ynones using DMF as dual synthon

Published:2020 Issue:48 Volume:56 Page:6488-6491
ISSN:1359-7345
Container-title:Chemical Communications
language:en
Short-container-title:Chem. Commun.

Author:

Ganesan Balaji¹²³⁴^ORCID,Govindan Karthick¹²³⁴^ORCID,Senadi Gopal Chandru⁵⁶⁷⁸⁹^ORCID,Kandasamy Mohanraj¹²³⁴^ORCID,Lin Wei-Yu¹²³⁴¹⁰^ORCID

Affiliation:

1. Department of Medicinal and Applied Chemistry

2. Kaohsiung Medical University

3. Taiwan

4. Republic of China

5. Department of Chemistry

6. Faculty of Engineering and Technology

7. SRM Institute of Science and Technology

8. Chennai-603203

9. India

10. Department of Medical Research

Abstract

The utilization of DMF as a dual synthon to serve as a methine source to introduce C2 carbon and nitrogen source to incorporate amino functionality in the 4^th position of quinoline under Cu-catalysis.

Funder

Ministry of Science and Technology, Taiwan

Kaohsiung Medical University

Publisher

Royal Society of Chemistry (RSC)

Subject

Materials Chemistry,Metals and Alloys,Surfaces, Coatings and Films,General Chemistry,Ceramics and Composites,Electronic, Optical and Magnetic Materials,Catalysis

Link

http://pubs.rsc.org/en/content/articlepdf/2020/CC/D0CC03033C

Reference44 articles.

1. A review on diverse heterocyclic compounds as the privileged scaffolds in antimalarial drug discovery

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5. Assembly of 4-Aminoquinolines via Palladium Catalysis: A Mild and Convenient Alternative to SNAr Methodology

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