Enantioselective construction of tricyclic pyrrolidine-fused benzo[b]thiophene 1,1-dioxide derivatives via copper(i)-catalyzed asymmetric 1,3-dipolar cycloaddition-Reference-Cited by-同舟云学术

Enantioselective construction of tricyclic pyrrolidine-fused benzo[b]thiophene 1,1-dioxide derivatives via copper(i)-catalyzed asymmetric 1,3-dipolar cycloaddition

Published:2017 Issue:12 Volume:4 Page:2343-2347
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Deng Hua¹²³⁴,He Fu-Sheng¹²³⁴,Li Cong-Shan¹²³⁴,Yang Wu-Lin¹²³⁴,Deng Wei-Ping¹²³⁴^ORCID

Affiliation:

1. School of Pharmacy and Shanghai Key Laboratory of New Drug Design

2. East China University of Science and Technology

3. Shanghai 200237

4. People's Republic of China

Abstract

A facile Cu(i)-catalyzed asymmetric 1,3-dipolar cycloaddition is developed, affording chiral tricyclic pyrrolidine-fused benzo[b]thiophene derivatives in excellent diastereo- and enantioselectivities.

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2017/QO/C7QO00640C

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4. Enantioselective Photocyclization of 2-Arylthio-3-methylcyclohexen-1-ones to Dihydrobenzothiophene Derivatives in an Inclusion Crystal with an Optically Active Host

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