Radical cascade synthesis of azoles via tandem hydrogen atom transfer-Reference-Cited by-同舟云学术

Radical cascade synthesis of azoles via tandem hydrogen atom transfer

Published:2020 Issue:9 Volume:11 Page:2479-2486
ISSN:2041-6520
Container-title:Chemical Science
language:en
Short-container-title:Chem. Sci.

Author:

Chen Andrew D.¹²³⁴,Herbort James H.¹²³⁴,Wappes Ethan A.¹²³⁴,Nakafuku Kohki M.¹²³⁴,Mustafa Darsheed N.¹²³⁴,Nagib David A.¹²³⁴^ORCID

Affiliation:

1. Department of Chemistry and Biochemistry

2. The Ohio State University

3. Columbus

4. USA

Abstract

A radical cascade enables rapid, modular access to five-membered heteroarenes, including oxazoles and imidazoles, through a regio- and chemo-selective β C–H bis-functionalization.

Funder

Alfred P. Sloan Foundation

National Institute of General Medical Sciences

Division of Chemistry

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/SC/C9SC06239D

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3. Mitigating Heterocycle Metabolism in Drug Discovery

4. Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design

5. Chemistry of oxazoles

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