Diastereoselective synthesis of highly functionalized polycyclic benzosultams via tandem cyclisations of cyclic N-sulfonylimines with in situ generated Huisgen 1,4-dipoles
Author:
Affiliation:
1. College of Life Science and Bio-engineering
2. Beijing University of Technology
3. Beijing 100124
4. P. R. China
Abstract
The tandem cycloadditions of cyclic N-sulfonylimines with in situ generated Huisgen 1,4-dipoles underwent readily, and delivered 1,2,3,4-tetrahydropyrimidine-fused benzosultams in acceptable chemical yields with excellent diastereoselectivities.
Funder
Beijing Municipal Commission of Education
Publisher
Royal Society of Chemistry (RSC)
Subject
General Chemical Engineering,General Chemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2016/RA/C6RA12771A
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