Rh-Catalyzed C–H activation/intramolecular condensation for the construction of benzo[f]pyrazolo[1,5-a][1,3]diazepines-Reference-Cited by-同舟云学术

Rh-Catalyzed C–H activation/intramolecular condensation for the construction of benzo[f]pyrazolo[1,5-a][1,3]diazepines

Published:2020 Issue:15 Volume:18 Page:2893-2901
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Ning Yi¹²³⁴⁵,He Xinwei¹²³⁴⁵^ORCID,Zuo Youpeng¹²³⁴⁵,Wang Jian¹²³⁴⁵^ORCID,Tang Qiang¹²³⁴⁵,Xie Mengqing¹²³⁴⁵,Li Ruxue¹²³⁴⁵,Shang Yongjia¹²³⁴⁵^ORCID

Affiliation:

1. Key Laboratory of Functional Molecular Solids

2. Ministry of Education

3. Anhui Laboratory of Molecule-Based Materials (State Key Laboratory Cultivation Base)

4. College of Chemistry and Materials Science

5. Anhui Normal University

Abstract

A novel and mild Rh(iii)-catalyzed cascade C–H activation/intramolecular condensation of 1-aryl-1H-pyrazol-5-amines with cyclic 2-diazo-1,3-diketones for the synthesis of various important benzo[f]pyrazolo[1,5-a][1,3]diazepines has been developed.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Anhui Province

Anhui Normal University

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/OB/D0OB00382D

Reference71 articles.

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