Synthesis, antiribosomal and antibacterial activity of 4′-O-glycopyranosyl paromomycin aminoglycoside antibiotics-Reference-Cited by-同舟云学术

Synthesis, antiribosomal and antibacterial activity of 4′-O-glycopyranosyl paromomycin aminoglycoside antibiotics

Published:2014 Issue:8 Volume:5 Page:1179-1187
ISSN:2040-2503
Container-title:MedChemComm
language:en
Short-container-title:Med. Chem. Commun.

Author:

Chen Weiwei¹²³⁴,Matsushita Takahiko¹²³⁴,Shcherbakov Dimitri⁵⁶⁷⁸,Boukari Heithem⁵⁶⁷⁸,Vasella Andrea⁹¹⁰¹¹⁸,Böttger Erik C.⁵⁶⁷⁸,Crich David¹²³⁴

Affiliation:

1. Department of Chemistry

2. Wayne State University

3. Detroit

4. USA

5. Institut für Medizinische Mikrobiologie

6. Universität Zürich

7. 8006 Zürich

8. Switzerland

9. Laboratorium für Organische Chemie

10. ETH Zürich

11. 8093 Zürich

Abstract

4′-O-Glycopyranosylation of the aminoglycoside paromomycin affects differentially the inhibition of prokaryotic and eukaryotic ribosomes and influences antibacterial activity against MRSA.

Publisher

Royal Society of Chemistry (RSC)

Subject

Pharmaceutical Science,Biochemistry,Drug Discovery,Molecular Medicine,Pharmacology,Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2014/MD/C4MD00119B

Reference41 articles.

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2. Aminoglycoside Antibiotics in the 21st Century

3. The Future of Aminoglycosides: The End or Renaissance?

4. Versatility of Aminoglycosides and Prospects for Their Future

5. Synthesis and Spectrum of the Neoglycoside ACHN-490

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