Galacto configured N-aminoaziridines: a new type of irreversible inhibitor of β-galactosidases
Author:
Affiliation:
1. Medicinal Chemistry Laboratory (MedChemLab)
2. Departament de Química Biomèdica
3. Institut de Química Avançada de Catalunya (IQAC–CSIC)
4. Barcelona
5. Spain
6. NMR Unit
Abstract
N-Aminoaziridines are potent irreversible inhibitors of galactosidases.
Publisher
Royal Society of Chemistry (RSC)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
http://pubs.rsc.org/en/content/articlepdf/2015/OB/C5OB00532A
Reference54 articles.
1. Glycosidase inhibitors: update and perspectives on practical use
2. D. P. Kasbekar and K.McCluskey, Neurospora: Genomics and Molecular Biology, 2013, Caister Academic Press
3. Glycosidase activities in bovine milk over lactation
4. Physiological roles of plant glycoside hydrolases
5. Sugar-mimic glycosidase inhibitors: natural occurrence, biological activity and prospects for therapeutic application
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